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MANDELATE RACEMASE: INSIGHTS INTO SUBSTRATE TOLERANCE, NOVEL INHIBITOR-BINDING MODES, AND THE ROLE OF BINDING DETERMINANTS
(2016-12-05)
Mandelate racemase (MR) is a useful model for studying the enzyme-catalyzed abstraction of an α-proton from carbon acid substrates with high pKa values. MR, an archetype of enolase superfamily, uses the Brønsted acid-base ...